Iron Sucrose — Active Pharmaceutical Ingredient

Iron Sucrose is an active pharmaceutical ingredient found in 2 FDA-approved drug products. Forms: INJECTABLE. Routes: INTRAVENOUS.

This content is for informational purposes only. Always consult a healthcare professional.

Iron Sucrose (2 brand names, 1 dosage form, 1 route)

Available dosage forms: INJECTABLE.

Routes of administration: INTRAVENOUS.

Brand Names

  • IRON SUCROSE
  • VENOFER

Indications and Usage

Iron Sucrose Injection is indicated for the treatment of iron deficiency anemia (IDA) in patients with chronic kidney disease (CKD).

Contraindications

Known hypersensitivity to Iron Sucrose Injection

Adverse Reactions

The following clinically significant adverse reactions are described elsewhere in the labeling:• Hypersensitivity Reactions [ see Warnings and Precautions (5.1) ] • Hypotension [ see Warnings and Precautions (5.2) ] • Iron Overload [ see Warnings and Precautions (5.3) ]

Drug Interactions

Iron Sucrose Injection may reduce the absorption of concomitantly administered oral iron preparations.

Mechanism of Action

Iron Sucrose Injection is an aqueous complex of poly-nuclear iron (III)-hydroxide in sucrose. Following intravenous administration, Iron Sucrose Injection is dissociated into iron and sucrose and the iron is transported as a complex with transferrin to target cells including erythroid precursor cells. The iron in the precursor cells is incorporated into hemoglobin as the cells mature into red blood cells.

Overdosage

No data are available regarding overdosage of Iron Sucrose Injection in humans. Excessive dosages of Iron Sucrose Injection may lead to accumulation of iron in storage sites potentially leading to hemosiderosis. Do not administer Iron Sucrose Injection to patients with iron overload [see Warnings and Precautions (5.3)]. Iron Sucrose Injection is not dialyzable through CA210 (Baxter) High Efficiency or Fresenius F80A High Flux dialysis membranes. Toxicities in single-dose studies in mice and rats, at intravenous iron sucrose doses up to 8 times the maximum recommended human dose based on body surface area, included sedation, hypoactivity, pale eyes, bleeding in the gastrointestinal tract and lungs, and mortality.

⚠ Caution
Medical Disclaimer: This information is for educational purposes only. Always consult a healthcare professional before taking any medication.