Bepotastine Besilate — Active Pharmaceutical Ingredient

Bepotastine Besilate is an active pharmaceutical ingredient found in 2 FDA-approved drug products. Forms: SOLUTION/DROPS, SOLUTION. Routes: OPHTHALMIC.

This content is for informational purposes only. Always consult a healthcare professional.

Bepotastine Besilate (2 brand names, 2 dosage forms, 1 route)

Available dosage forms: SOLUTION/DROPS, SOLUTION.

Routes of administration: OPHTHALMIC.

Brand Names

  • BEPOTASTINE BESILATE
  • BEPREVE

Indications and Usage

Bepotastine besilate ophthalmic solution, 1.5% is a histamine H1 receptor antagonist indicated for the treatment of itching associated with signs and symptoms of allergic conjunctivitis.

Dosage and Administration

Instill one drop of bepotastine besilate ophthalmic solution into the affected eye(s) twice a day. Remove contact lenses prior to instillation of bepotastine besilate ophthalmic solution.

Contraindications

Bepotastine besilate ophthalmic solution is contraindicated in patients with a history of hypersensitivity reactions to bepotastine or any of the other ingredients [see Adverse Reactions (6.2)].

Mechanism of Action

Bepotastine is a topically active, direct H1-receptor antagonist and an inhibitor of the release of histamine from mast cells.

⚠ Caution
Medical Disclaimer: This information is for educational purposes only. Always consult a healthcare professional before taking any medication.